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NITRATONG Nitroxinil Injection 34%

Short Tlhaloso:

Sebopeho mong le e mong 1ml na Nitroxynil 340mg le Excipients qsto 1ml. TLHALOSO E ke bo bofubelu injectable tharollo. lebitso Generic: Nitroxynil ente 34%. Lebitso cha: Nitrodox 34 lik'hemik'hale Name: Lodine-2-hydroxi-4-nitro-5-benzonitrile (cyano4-a iodine litareng e, 2, nitro-6phenol) lik'hemik'hale Sebopeho: Mol Weight: 290,02 CAS No: 1689-89-0 CLNICAL PHARMACOLOGY Parmacodynamics : Nitrodox 34 ke nitrate sehlahisoa tloha metsoako benzene le hlahisa le phello e flukicide le e atisa ho sebelisoa le ...


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Sebopeho

E mong le e 1ml na Nitroxynil 340mg le Excipients qsto 1ml.

 

TLHALOSO

Ke bo bofubelu injectable tharollo.

Lebitso Generic: Nitroxynil ente 34%.

Lebitso cha: Nitrodox 34

Lik'hemik'hale Name: Lodine-2-hydroxi-4-nitro-5-benzonitrile (cyano4-a iodine litareng e, 2, nitro-6phenol)

Lik'hemik'hale Sebopeho:

Mol Weight: 290,02 CAS No: 1689-89-0

 

CLNICAL PHARMACOLOGY

Parmacodynamics:

Nitrodox 34 ke nitrate sehlahisoa tloha metsoako benzene le hlahisa le phello e flukicide le e atisa ho sebelisoa le 'ngoe le a manyenyane ho fetisisa ho tloha nitrate tsohle trematocides sehlahisoa. The mochine oa ketso e lumellana ho hema metabolism tshitsiso tsa helminth e, thibela ho hlahisa matla ka hore phosphorylation mitochondrial oxidative. Nitrodox 34 ka sitisang ho sebelisa itšoare ka oxide e-phokotso ya adenosine diphosphate (ATP) tlhahiso. Ka mor'a ho sebelisa mehloli eohle ea eona mahlahahlaha le likokoana-hloko shoa ka lebaka la ho bolaoa ke tlala.

 

Nitrodox 34 hape e etsa hore detachment scolex tsa mucosa mala le proglottid proximal tsa cestode ena.

 

Lithuto tsa ka hlokomela le Nitrodox 34 bontša hore maemo e atlehang ea mali li ile tsa fihla ka mor'a lihora tse 5 tsa tsamaiso ea lithethefatsi le ka litlhōrō tse lebetsoeng le ka mor'a lihora tse 12, ka mosebetsi monyako matsatsing 30 hore maximizes bohato lona antiparasitic.

 

Pharmacokinetics:

Ho na le ka ho hlokomela hore e amahanngoa ka matla ho liprotheine plasmatic bakopitsi ho kabo lona ho lisele tse ba le ho ntsha lona lieha ya phelang. The biotransformation le hlaha ka pampitšana gastrointestinal le sebete. The Nitrodox 34 le metabolites lona ba felisoa ke masi ka tsela e bile.

 

E etsa tlhahiso ea hore e sebetsang sebakeng sa hae inhibiting phosphorylation le oxidative. Ho ka etsahala ho netefatsa liphello tsa eona tse fetang Fasciola gigantica ka maemo laboratoring, ka mor'a ho eketsa 20 mg, / ml tse ka vitro, e bitsang setopong se hang-hang ya pelehi mesifa, ho etsa ba nahana hore liketso tsa ka blocker neuromuscular, ka lebaka la ena ea parasite hlokahala shoele litho le le khaello matla.

Nitrodox 34 e sebediswa ke tsela parenteral hobane ka koko ho ne a tla utloa e le phokotso bokgoni; e lebetsoeng le maemo plasmatic di fumana pakeng tsa metsotso e 30 le 60 le bophelo li bolela'ng ke matsatsi a 8; ea excretion le hlaha ka moroto matsatsing 30 hoo e ka bang.

 

ho bonahala

Nitrodox 34 e bontša bakeng sa taolo ya Fasciolosis (larval le batho ba baholo sethaleng) ile a etsa hore ke Fasciola hepatica le F. gigantica; gastrointestinal parasitism bakoang ke Haemonchus spp., Bunostomum spp., Oesophagostomum spp., Oestrus spp. ka likhomo, linku, lipoli le kamele, hammoho le

Ancylostoma spp. le Uncinaria spp.in lintja.

 

phofu ya diphoofolo

Nitrodox 34 e ntshetswa pele le diteko tsa ho e sebelisa ka likhomo, linku, lipoli, kamele le lintja.

 

Litekanyetso li behoa le taolo

Subcutaneous tsela feela.

The litekanyetso li behoa Standard ke 10mg ka 1 lik'hilograma bodyweight (= 1.5 di ml Nitrodox 34 / 50kg BW).

 

Likhomo, Sheep, Pōli, likamele le Dogs:

1ml mong le e mong 50kg tsa boima ba 'mele khahlanong le Fasciola hepatica le F.gigantica.

1.5 di ml mong le e mong boima ba lik'hilograma tse 50 tsa boima ba 'mele khahlanong le Haemochus contortus, Oesophagostomum spp., Bunostomum spp., Ancylostoma caninum le Uncinatia spp.

2.0 di ml mong le e mong boima ba lik'hilograma tse 50 tsa boima ba 'mele ka maemo a ho a hlobaetsang haholo Fasciolosis le Oestrosis ka le linku tsa ka (Oestrus ovis).

 

Lehlakoreng LIPHELLO

A ruruha hanyenyane 'na la bonahala ka site ya inoculation, e leng tla nyamela ka matsatsi a' maloa.

 

Mehato LE TEMOSO

1. feela lethal dose likhomo ka nako e omme.

2. U se ke ua kopanya ea ente e tšoanang kapa setshelo le ntho leha e le efe e fapaneng ho sehlahiswa.

The lik'hontheinara le masalla efe kapa efe ya sehlahiswa lokela ho felisoa ka tsela e sireletsehileng (lepato kapa incineration).

3. Ho sebelisa ka mefuta e meng e fetang matla e sa kgothaletswa.

4. E ka sebediswa e jele efe kapa efe ya ho ima (Leha ho le joalo, ka boraro ea ho qetela, sehlahiswa tlameha ho khona ka hloko haholo tlas'a tlhokomelo litsebi); ha ho ama tsoalo, emara kapa sebopeho lesea, 'me ha ho ama tshebetso ho ikatisa ya stallions.

5. Tabeng ea botahoa, le 'ne le mamello sebakeng se batang le laola dextrose ke tsela endovenous.

6. Ka Ha a e-ja, ho hlatsoa molomo le kopo thuso ho veterinarian ena.

7. E-ba hlokolosi ba likoloi nkente ka phoso. Batla ngakeng tabeng ea ente ka phoso.

 

a khaotsa ho tsuba NAKO

Nama: matsatsi a 30. Lebese: matsatsi a 5. Lethal dose likhomo feela ka nako e omme.

 

bonnete

lilemo tse 2

 

PRESENTAION

Nitrodox 34 e fumaneha ka botlolo ea 100ml, le 250ml.

 

Storage

Boloka a pholile, e omeletseng le lefifi sebaka.


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